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Inhibitors

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CAS:1231929-97-7
Molecular Formula:C27H32F2N8
N-(5-((4-Ethylpiperazin-1-yl)Methyl)Pyridin-2-yl)-5-Fluoro-4-(4-Fluoro-1-Isopropyl-2-Methyl-1H-Benzo[d]Imidazol-6-yl)Pyrimidin-2-Amine
Brief Introduction
Abemaciclib is an oral cyclin dependent kinase CDK4 / 6 inhibitor
CAS:104121-92-8
Molecular Formula:C30H50O5
2-(3-Hydroxypropoxy)-1,25-Dihydroxyvitamin D3; (1R,Z)-5-((E)-2-((1R,7aR)-1-((R)-6-Hydroxy-6-Methylheptan-2-yl)-7a-Methylhexahydro-1H-Inden-4(2H)-Ylidene)Ethylidene)-2-(3-Hydroxypropoxy)-4-Methylenecyclohexane-1,3-diol1Alpha,25-Dihydroxy-2beta-(3-Hydroxypropoxy)Vitamin D3; (1S,2S,3S,5Z)-5-[(2E)-2-[(1R,3aS,7aR)-1-[(2R)-6-Hydroxy-6-Methylheptan-2-yl]-7a-Methyl-2,3,3a,5,6,7-Hexahydro-1H-Inden-4-Ylidene]Ethylidene]-2-(3-Hydroxypropoxy)-4-Methylidenecyclohexane-1,3-diol
Brief Introduction
Eldecalcitol is an active vitamin D3 derivative, which acts on human osteoclast precursor cells and inhibits the formation of osteoclasts.
CAS:917389-32-3
Molecular Formula:C29H28F4N4O4
AIC246; CS-2799; MK-8828; UNII-1H09Y5WO1F; (4S)-8-Fluoro-3,4-Dihydro-2-[4-(3-Methoxyphenyl)-1-Piperazinyl]-3-[2-Methoxy-5-(Trifluoromethyl)Phenyl]-4-Quinazolineacetic acid; -Quinazolineacetic acid, 8-Fluoro-3,4-Dihydro-2-[4-(3-Methoxyphenyl)-1-Piperazinyl]-3-[2-Methoxy-5-(Trifluoromethyl)Phenyl]-, (4S)-
Brief Introduction
Letimovir is a novel anti CMV compound, which targets the virus terminal enzyme complex. Viruses resistant to DNA polymerase inhibitors also have activity.
CAS:906673-24-3
Molecular Formula:C14H10BNO3
4-((1-Hydroxy-1,3-Dihydrobenzo[c][1,2]Oxaborol-5-yl)oxy)Benzonitrile; 5-(4-Cyanophenoxy)-2,3-Dihydro-1-Hydroxy-2,1-Benzoxaborole; Eucrisa; 4-[(1-Hydroxy-3H-2,1-Benzoxaborol-5-yl)oxy]Benzonitrile; 4-(1-Hydroxy-1,3-Dihydrobenzo[c][1,2]Oxaborol-5-Yloxy)Benzonitrile; 4-[(1,3-Dihydro-1-Hydroxy-2,1-Benzoxaborol-5-yl)oxy]Benzonitrile
Brief Introduction
Crisaborole is a PDE4 inhibitor. PDE4 activity is increased in circulating inflammatory cells in patients with atopic dermatitis. PDE4 is a very core regulatory point for the production of inflammatory cytokines in atopic dermatitis, mainly through the degradation of cyclic adenosine monophosphate.
CAS:1622902-68-4
Molecular Formula:C14H21N5O2S
PF-04965842; 1-Propanesulfonamide, N-[cis-3-(Methyl-7H-Pyrrolo[2,3-d]Pyrimidin-4-Ylamino)Cyclobutyl]-; N-[cis-3-[Methyl(7H-Pyrrolo[2,3-d]Pyrimidin-4-yl)Amino]Cyclobutyl]Propane-1-Sulfonamide
Brief Introduction
PF-04965842 (Abrotinib) is a small molecule JAK inhibitor that is orally administered once daily and can selectively inhibit JAK1. JAK1 inhibitors can participate in regulating various cytokines in the pathology of atopic dermatitis.
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