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Inhibitors

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CAS:171599-83-0
Molecular Formula:C28H38N6O11S
Sildenafil Citrate Salt; 5-[2-Ethoxy-5-(4-Methylpiperazin-1-Yl)Sulfonylphenyl]-1-Methyl-3-Propyl-4H-Pyrazolo[4,3-D]Pyrimidin-7-One,2-Hydroxypropane-1,2,3-Tricarboxylic Acid; Viagra,Revatio; Viagra, Sildenafil Citrate; 1-[[3-(4,7-Dihydro-1-Methyl-7-Oxo-3-Propyl-1H-Pyrazolo[4,3-D]Pyrimidin-5-Yl)-4-Ethoxyphenyl]Sulfonyl]-4-Methylpiperazine Citrate Salt; 5-[2-Ethoxy-5-(4-Methylpiperazin-1-Yl)Sulfonylphenyl]-1-Methyl-3-Propyl-4H-Pyrazolo[5,4-E]Pyrimidin-7-One Citrate Salt; 1-[[3-(6,7-Dihydro-1-Methyl-7-Oxo-3-Propyl-1H-Pyrazolo[4,3-D]Pyrimidin-5-Yl)-4-Ethoxyphenyl]Sulfonyl]-4-Methylpiperazine, 2-Hydroxy-1,2,3-Propanetricarboxylate; 5-[2-Ethoxy-5-[(4-Methyl-Piperazin-1-Yl)Sulfonyl]Phenyl]-1,6-Dihydro-1-Methyl-3-Propyl-7H-Pyrazolo[4,3-D]Pyrimidin-7-One Citrate
Brief Introduction
Sildenafil citrate, a selective 5-phosphodiesterase inhibitor, enhances nitric oxide dependent pulmonary vasodilation mediated by cyclic guanosine monophosphate by inhibiting the decomposition of cyclic guanosine monophosphate. In addition to direct dilation of pulmonary vessels, it can also prevent or reverse vascular remodeling. It is used for impotence patients with erectile dysfunction.
CAS:23672-07-3
Molecular Formula:C15H23N3O4S
(S)-(-)-5-(Aminosulfonyl)-N-[(1-Ethyl-2-Pyrrolinyl)Methyl]; S(-)-Sulpiride Dopamine D1 Antagonis; Benzamide, 5-(Aminosulfonyl)-N-[(1-Ethyl-2-Pyrrolidinyl)Methyl]-2-Methoxy-, (S)-; Benzamide, 5-(Aminosulfonyl)-N-[[(2S)-1-Ethyl-2-Pyrrolidinyl]Methyl]-2-Methoxy- (9Ci); L-Sulpiride; (S)-(-)-N-((1-Ethyl-2-Pyrrolidinyl)Methyl)-5-Sulfamoyl-O-Anisamide 5-(Aminosulfonyl)-N-((1-Ethyl-2-Pyrrolidinyl)Methyl)-2-Methoxy-Benzamid ( S-(-)-Benzamid
Brief Introduction
This product is a levorotator of sulpiride. They have similar effects and uses. They are used as antipsychotics and prokinetic agents.
CAS:364782-34-3
Molecular Formula:C22H23ClF3N
Mimpara; Sensipar; Cinacalcet Hcl; (R)-N-(1-(Naphthalen-1-Yl)Ethyl)-3-(3-(Trifluoromethyl)Phenyl)Propan-1-Amine Hydrochloride; (Ar)-A-Methyl-N-[3-[3-(Trifluoromethyl)Phenyl)Propyl]-1-Napthalenemethanamine Hydrochloride; N-[(1R)-1-Naphthalen-1-Ylethyl]-3-[3-(Trifluoromethyl)Phenyl]Propan-1-Amine Hydrochloride; -Naphthalenemethanamine, .Alpha.-Methyl-N-[3-[3-(Trifluoromethyl)Phenyl]Propyl]-, Hydrochloride
Brief Introduction
Cinacalcet Hydrochloride is a specific drug for controlling hyperparathyroidism and inhibiting parathyroid hormone PTH.
CAS:439081-18-2
Molecular Formula:C24H25ClFN5O3
Tovok; BIBW2992; (S)-N-(4-((3-Chloro-4-Fluorophenyl)Amino)-7-((Tetrahydrofuran-3-Yl)Oxy)Quinazolin-6-Yl)-4-(Dimethylamino)But-2-Enamide; 2-Butenamide, N-[4-[(3-Chloro-4-Fluorophenyl)Amino]-7-[[(3S)-Tetrahydro-3-Furanyl]Oxy]-6-Quinazolinyl]-4-(Dimethylamino)-; (E/Z)-Afatinib; Afatinib Cis-Trans Isomer; Bibw-2292
Brief Introduction
Afatinib is an aminocrotonyl amino substituted quinazoline derivative used to treat cancers and diseases of respiratory tract, lung, gastrointestinal tract, bile duct and gallbladder.
CAS:503612-47-3
Molecular Formula:C25H25N5O4
1-(4-Methoxyphenyl)-7-Oxo-6-[4-(2-Oxopiperidin-1-Yl)Phenyl]-4,5-Dihydropyrazolo[3,4-C]Pyridine-3-Carboxamide; Eliquis; Unii-3Z9Y7Uwc1J; Bms-562247-01; Bms-562247
Brief Introduction
Apixaban (inn, trade name eliquis) is an anticoagulant used to prevent venous thromboembolism and atrial fibrillation stroke. It is a direct factor Xa inhibitor. Apixaban has been listed in Europe since May 2011. The drug was developed by a joint venture between Pfizer and Bristol Myers Squibb.
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