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Inhibitors

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CAS:74103-07-4
Molecular Formula:C19H24N2O6
2-Amino-2-(Hydroxymethyl)Propane-1,3-Diol,5-Benzoyl-2,3-Dihydro-1H-Pyrrolizine-1-Carboxylic Acid; Rac Ketorolac Tromethamine Salt; Ketorolac Tris Salt; Toradol; Acular
Brief Introduction
Ketorolac tromethamine is an alcohol organic compound. Its biological activity is related to L-S (-) and can inhibit prostaglandin biosynthesis.
Hainan Zhuoke Pharmaceutical Co., Ltd.
CNY 100 Million
19980m²
Less Than 50 People
CRO CRO
Product Photo Specification Grade Max Capacity Certificates Package
YBH03222006,CP Pharm Grade - -
10kg / Fibre Drum
Main products:
Ketorolac Tromethamine /Sulpiride /Diatrizoic Acid Dihydrate /Meglumine /Mycophenolate Mofetil /Aztreonam /Cefamandole Nafate /Creatine Phosphate Disodium Salt
CAS:868540-17-4
Molecular Formula:C40H57N5O7
(2S)-4-Methyl-N-[(2S)-1-[[(2S)-4-Methyl-1-[(2R)-2-Methyloxiran-2-Yl]-1-Oxopentan-2-Yl]Amino]-1-Oxo-3-Phenylpropan-2-Yl]-2-[[(2S)-2-[(2-Morpholin-4-Ylacetyl)Amino]-4-Phenylbutanoyl]Amino]Pentanamide; Kyprolis; Unii-72X6E3J5Ar; Carfilzomib (PR-171); PR-171
Brief Introduction
Carfilzomib is a proteasome inhibitor. Proteasome can decompose proteins that are damaged or no longer needed, thus playing an important role in cell function and growth.
CNY 39.8 Million
19980m²
100-500 People
CRO CRO
Product Photo Specification Grade Max Capacity Certificates Package
98% Pharm Grade - -
25kg / Fibre Drum
Main products:
Carfilzomib /Relugolix /Ixazomib Citrate /Apalutamide /Avatrombopag /Fulvestrant /Lenvatinib Mesylate /Ruxolitinib Phosphate /Roxadustat /Brivaracetam
CAS:1051375-16-6
Molecular Formula:C20H19F2N3O5
(4R,12As)-N-(2,4-Difluorobenzyl)-7-Hydroxy-4-Methyl-6,8-Dioxo-3,4,6,8,12,12A-Hexahydro-2H-Pyrido[1',2':4,5]Pyrazino[2,1-B][1,3]Oxazine-9-Carboxamide; S/Gsk1349572; Gsk 1349572; Tivicay; Dtg; Dolutegravir Api; Dolutegravir (Gsk1349572); 2H-Pyrido[1',2'
Brief Introduction
Dolutegravir (DTG) is an FDA-approved drug for the treatment of HIV infection. Dolutegravir is an integrase inhibitor. Known as S/GSK1349572 or just "572" the drug is marketed as Tivicay by GlaxoSmithKline (GSK). In February, 2013 the Food and Drug Administration announced that it would fast track dolutegravir's approval process. On August 13, 2013, dolutegravir was approved by the FDA. On November 4, 2013, dolutegravir was approved by Health Canada. On January 16, 2014, Tivicay was approved by the European Commission for use throughout the European Union.
CNY 22 Million
49950m²
100-500 People
CRO CRO
Product Photo Specification Grade Max Capacity Certificates Package
WHO Pharm Grade - -
25kg / Fibre Drum
Main products:
Dolutegravir /Sodium 4-Aminosalicylate Dihydrate /Metoclopramide Hydrochloride /Ambroxol Hydrochloride /Ethacridine Lactate Monohydrate /Metoclopramide /Metaraminol Bitartrate /Moxifloxacin Hydrochloride /Sacubitril /2-Chloro-4-Nitrobenzoic Acid /Bictegravir /Methyl 4-Acetamido-2-Methoxybenzoate /Methyl 4-Acetamido-5-Chloro-2-Methoxybenzoate /Bromhexine Hydrochloride /4-Aminosalicylic Acid
CAS:1092939-17-7
Molecular Formula:C17H21N6O4P
3R)-Cyclopentyl-3-[4-(7H-Pyrrolo[2,3-d]Pyrimidin-4-yl)Pyrazol-1-yl]Propionitrile Phosphate; (R)-3-(4-(7H-Pyrrolo[2,3-d]Pyrimidin-4-yl)-1H-Pyrazol-1-yl)-3-Cyclopentylpropanenitrile Phosphate; Jakafi; Jakavi
Brief Introduction
Ruxolitinib phosphate is a potent JAK1/2 inhibitor with IC50 of 3.3 nM/2.8 nM, respectively, showing 130-fold selectivity over JAK3.
CNY 39.8 Million
19980m²
100-500 People
CRO CRO
Product Photo Specification Grade Max Capacity Certificates Package
99% Pharm Grade - -
25kg / Fibre Drum
Main products:
Ruxolitinib Phosphate /Relugolix /Carfilzomib /Ixazomib Citrate /Apalutamide /Avatrombopag /Fulvestrant /Lenvatinib Mesylate /Roxadustat /Brivaracetam
CAS:109581-93-3
Molecular Formula:C44H71NO13
Tacrolimus; Tacrolimus Hydrate; Prograf; Protopic; Tsukubaenolide Hydrate
Brief Introduction
Tacrolimus monohydrate (FK506 monohydrate) is a macrolide compound that binds to the FK506 binding protein (FKBP) to form a complex and inhibits calcineurin phosphatase, thereby inhibiting T lymphocyte signal transduction and IL-2 transcription. Has strong immunosuppressive properties.
USD 5 Million
50-100 People
Manufacturing Manufacturing
Product Photo Specification Grade Max Capacity Certificates Package
97% to 102% Pharm Grade 180 tons/year
1kg / Fibre Drum
98.0 % to 102.0% Pharm Grade 180 tons/year
1kg / Fibre Drum
Main products:
Tacrolimus Monohydrate
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