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Inhibitors

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CAS:1609392-27-9
Molecular Formula:C20H19D3N8O3
BMS-986165; Tyk2-IN-4; Sotyktu; 6-(Cyclopropanecarboxamido)-4-((2-Methoxy-3-(1-Methyl-1H-1,2,4-Triazol-3-yl)Phenyl)Amino)-N-(Methyl-d3)Pyridazine-3-Carboxamide; Deucravacitinib (BMS-986165)
Brief Introduction
Deucravacitinib is a Tyrosine Kinase 2 Inhibitor. The mechanism of action of deucravacitinib is as a Tyrosine Kinase 2 Inhibitor.
CAS:14680-51-4
Molecular Formula:C21H26N4O3
Benzimidazole, 1-(2-(Diethylamino)Ethyl)-2-(p-Methoxybenzyl)-5-Nitro-; N,N-Diethyl-2-((4-Methoxyphenyl)Methyl)-5-Nitro-1H-Benzimidazole-1-Ethanamine; N,N-Diethyl-2-[2-[(4-Methoxyphenyl)Methyl]-5-Nitrobenzimidazol-1-yl]Ethanamine; 1H-Benzimidazole-1-Ethanamine, N,N-Diethyl-2-((4-Methoxyphenyl)Methyl)-5-Nitro-; N,N-Diethyl-2-[(4-Methoxyphenyl)Methyl]-5-Nitro-1H-Benzimidazole-1-Ethanamine; 1-(2-Diethylaminoethyl)-2-(p-Methoxybenzyl)-5-Nitro-1H-Benzimidazole; N,N-Diethyl-2-(2-(4-Methoxybenzyl)-5-Nitro-1H-Benzimidazol-1-yl)Ethan-1-Amine
Brief Introduction
It is a pain relieving compound that has effects including analgesia, euphoria, and drowsiness.
CAS:1420477-60-6
Molecular Formula:C26H23N7O2
Calquence; Acalabrutiib; (S)-4-(8-Amino-3-(1-(but-2-Ynoyl)Pyrrolidin-2-yl)Imidazo[1,5-a]Pyrazin-1-yl)-N-(Pyridin-2-yl)Benzamide
Brief Introduction
Acalabrutinib is an experimental anti-cancer drug and a selective inhibitor of Bruton tyrosine kinase (BTK).
CAS:1110766-97-6
Molecular Formula:C29H32Cl2N2O5S
(E)-3-[2,6-Dichloro-4-[4-[3-[(S)-1-Hexyloxyethyl]-2-Methoxyphenyl]Thiazol-2-Ylcarbamoyl]Phenyl]-2-Methylacrylic acid
Brief Introduction
Lusutrombopag (Mulpleta, S-888711) is an orally bioavailable thrombopoietin (TPO) receptor agonist, currently being used in research for the treatment of chronic liver disease (CLD).
CAS:1422144-42-0
Molecular Formula:C30H35N3O9S2
AR-13324 (Mesylate); Benzoic acid,2,4-Dimethyl-,(4-((1S)-1-(Aminomethyl)-2-(6-Isoquinolinylamino)-2-Oxoethyl)Phenyl)Methyl Ester,Methanesulfonate (1:2); Netarsudil Dimesylate; AR-13324; (4-((1S)-1-(Aminomethyl)-2-(Isoquinolin-6-Ylamino)-2-Oxoethyl)Phenyl)Methyl 2,4-Dimethylbenzoate,Dimethanesulfonate
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