A partial adrenergic agonist with functional beta 1-receptor specificity and inotropic effect. It is effective in the treatment of acute CARDIAC FAILURE, postmyocardial infarction low-output syndrome, SHOCK, and reducing ORTHOSTATIC HYPOTENSION in the SHY-RAGER SYNDROME.

Aclacinomycin A

MSDS

CAS:57576-44-0

Molecular Formula:C42H53NO15

Alias

More Information

Aclacur; Aclarublcin; Aclacin; Jaclacin; Acm; Aclarubicin; Aelacinon; Ma144-A1; Aclaplastin; Aclarubicine; Aclarubicinum

Brief Introduction

The second generation of cyclocarcinoid antitumor antibiotics are cell cycle nonspecific drugs, which can inhibit the biosynthesis of DNA, RNA and protein. It has strong anticancer activity and can be administered VI. its toxicity to the heart is much lower than adriamycin, and has no obvious immunosuppressive and bone marrow inhibitory effects. Clinical use of its hydrochloride has a high degree of alleviation for acute leukemia, and is effective for uterine body cancer, liver cancer, gastrointestinal cancer, lung cancer, pancreatic cancer, ovarian cancer, and malignant lymphoma.

Fenobam

MSDS

CAS:57653-26-6

Molecular Formula:C11H11ClN4O2

Alias

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[3H]-Fenobam; N-3-Chlorophenyl-N'-(4,5-Dihydro-1-Methyl-4-Oxo-1H-Imidazol-2-Yl)Urea; 1-(3-Chlorophenyl)-3-(4,5-Dihydro-1-Methyl-4-Oxo-1H-Imidazol-2-Yl)Urea; N-(3-Chlorophenyl)-N'-(4,5-Dihydro-1-Methyl-4-Oxo-1H-Imidazole-2-Yl)Urea; 1-(3-Chlorophenyl)-3-(1-Methyl-4-Oxo-4,5-Dihydro-1H-Imidazol-2-Yl)Urea; Mcn-3377

Brief Introduction

Fenobam is a selective, orally active mGluR5 antagonist across the blood-brain barrier, which acts on allosteric regulatory sites (Kd values on rat and human recombinant mGlu5 receptors are 54 nm and 31 nm, respectively). Fenobam has reverse agonist activity, which blocks mGlu5 receptor activity with IC50 of 84 nm. Fenobam has anti anxiety activity.

Domperidone

CAS:57808-66-9

Molecular Formula:C22H24ClN5O2

Alias

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6-Chloro-3-[1-[3-(2-Oxo-3H-Benzimidazol-1-Yl)Propyl]Piperidin-4-Yl]-1H-Benzimidazol-2-One; Motilium; Nauzelin; Domperidonum

Brief Introduction

Domperidone is a benzimidazole compound, which has strong gastric motility and antiemetic effects. It can strengthen the tension of lower esophageal sphincter, prevent gastroesophageal reflux, enhance gastric peristalsis, promote gastric emptying, coordinate the movement of stomach and duodenum, inhibit nausea and vomiting, effectively prevent bile reflux and do not affect gastric juice secretion. This product is a peripheral dopamine receptor antagonist, which directly blocks the dopamine receptor in the gastrointestinal tract and promotes gastric motility. It can enhance the peristalsis of the esophagus and the tension of the lower esophageal sphincter. Because of its poor permeability to the blood-brain barrier and almost no antagonistic effect on dopamine receptors in the brain, it can eliminate the side effects of spirit and central nervous system.

Buserelina

MSDS

CAS:57982-77-1

Molecular Formula:C60H86N16O13

Alias

More Information

Buserelin; Etilamide; Busereline; Buserelinum; Metrelef; Buserelin (Inn); Tiloryth (Tn); Buserelin Acetate Salt; D-Ser-(Tbu)(Sup 6)-Lhrh-Ethylamide; (D-Ser(Tbu)(Sup 6)-Ea(Sup 10))-Lhrh; (D-Ser(Bu(Sup T)(Sup 6)))-Lh-Rh(1-9)Nonapeptide-Ethylamide; (D-Ser(Tbu)(Sup 6)-Ea(Sup 10))-Luteinizing Hormone-Releasing Hormone

Brief Introduction

Buserelin is a GnRH analogue. At the initial stage of use, it can increase the secretion of LH, FSH and sex hormone. After 1 ~ 2 weeks, it has the opposite effect, and the secretion of sex hormone can be reduced to the castration level. It is mainly used for prostate cancer, breast cancer and so on.

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