Appearance:White to grayish white crystalline powder
Synopsis:Tibolone is a tissue selective estrogen activity regulator (stairs), which is a synthetic steroid hormone. The hormone activity of tibolone itself is very weak, which mainly depends on the activity of local enzymes and tissue-specific metabolic mechanism, and plays different effects in different tissues. At present, I is mainly used in perimenopausal and postmenopausal women to alleviate vasomotor symptoms, improve urogenital atrophy symptoms, prevent bone loss, reduce the incidence of fracture and improve the quality of life Tibolone can stabilize the hypothalamic pituitary system in women after menopausal ovarian function decline.
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Summary
Tibolone is a tissue selective estrogen activity regulator (stairs), which is a synthetic steroid hormone. The hormone activity of tibolone itself is very weak, which mainly depends on the activity of local enzymes and tissue-specific metabolic mechanism, and plays different effects in different tissues. At present, I is mainly used in perimenopausal and postmenopausal women to alleviate vasomotor symptoms, improve urogenital atrophy symptoms, prevent bone loss, reduce the incidence of fracture and improve the quality of life Tibolone can stabilize the hypothalamic pituitary system in women after menopausal ovarian function decline.